List of drugs used to treat hypercholesterolemia, including various medications for hypercholesterolemia treatments. These medical treatments that are used to fight hypercholesterolemia are in alphabetical order, and may include pictures when available. If you are wondering, "What drugs are used to treat hypercholesterolemia?" consider that there are a variety of ways to treat hypercholesterolemia conditions. This hypercholesterolemia drug list includes the most common hypercholesterolemia medications and may include prescription drugs and nonprescription medications.Everything from Simvastatin to Atorvastatin is included on this list.